OG-L002

Catalog No. A13246

OG-L002是一种有效的特异性LSD1抑制剂,IC50为20 nM,分别比MAO-B和MAO-A表现出36倍和69倍的选择性。
Catalog Num A13246
M. Wt 261.75
Formula C15H15NO.HCl
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1357302-64-7
Synonyms OGL002, OG L002
SMILES CCOc1cc(ccc1Nc1ncc2c(n1)n(C)c1ccccc1c(=O)n2C)N1CCC(CC1)O
OG-L002是一种有效的特异性LSD1抑制剂,IC50为20 nM,分别比MAO-B和MAO-A表现出36倍和69倍的选择性。
Targets
LSD1 (Cell-free assay)
20 nM
In vitro (25°C) DMSO 41 mg/mL (181.99 mM)
Water Insoluble
Ethanol 17 mg/mL (75.45 mM)
In vivo 1% DMSO+30% polyethylene glycol+1% Tween 80 19 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 38.2 mL 191.02 mL 382.04 mL
0.5 mM 7.64 mL 38.2 mL 76.41 mL
1 mM 3.82 mL 19.1 mL 38.2 mL
5 mM 0.76 mL 3.82 mL 7.64 mL

*The above data is based on the productmolecular weight 261.75. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.