Anagliptin

Catalog No. A13529

Anagliptin是一种有效的选择性DPP-4抑制剂(IC50 = 3.8 nM);DPP-8和DPP-9的效力降低了10倍以上。
Catalog Num A13529
M. Wt 383.45
Formula C19H25N7O2
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 739366-20-2
Synonyms SK-0403
SMILES CC1=NN2C=C(C=NC2=C1)C(=O)NCC(C)(C)NCC(=O)N3CCC[C@H]3C#N
Anagliptin是一种有效的选择性DPP-4抑制剂(IC50 = 3.8 nM);DPP-8和DPP-9的效力降低了10倍以上。
In vitro DMSO 74 mg/mL (192.98 mM)
Water 19 mg/mL (49.54 mM)
Ethanol 74 mg/mL (192.98 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.08 mL 130.4 mL 260.79 mL
0.5 mM 5.22 mL 26.08 mL 52.16 mL
1 mM 2.61 mL 13.04 mL 26.08 mL
5 mM 0.52 mL 2.61 mL 5.22 mL

*The above data is based on the productmolecular weight 383.45. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.