GSK2801

Catalog No. A14015

GSK2801是BAZ2家族含溴结构域蛋白的强效抑制剂。
Catalog Num A14015
M. Wt 371.54
Formula C20H21NO4S
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1619994-68-1
Synonyms GSK-2801, GSK 2801
SMILES CCCOC1=CC2=C(C=C(N2C=C1)C(=O)C)C3=CC=CC=C3S(=O)(=O)C
GSK2801是BAZ2家族含溴结构域蛋白的强效抑制剂。
Targets
BAZ2B BAZ2A
136 nM(Kd)257 nM(Kd)
In vitro (25°C) DMSO Warmed: 67 mg/mL (180.37 mM)
Water Insoluble
Ethanol Warmed: 6 mg/mL (16.15 mM)
In vivo 0.5% CMC+1% Tween 80 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.92 mL 134.58 mL 269.15 mL
0.5 mM 5.38 mL 26.92 mL 53.83 mL
1 mM 2.69 mL 13.46 mL 26.92 mL
5 mM 0.54 mL 2.69 mL 5.38 mL

*The above data is based on the productmolecular weight 371.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.