GSK2801
Catalog No. A14015
GSK2801是BAZ2家族含溴结构域蛋白的强效抑制剂。
Catalog Num | A14015 |
---|---|
M. Wt | 371.54 |
Formula | C20H21NO4S |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1619994-68-1 |
Synonyms | GSK-2801, GSK 2801 |
SMILES | CCCOC1=CC2=C(C=C(N2C=C1)C(=O)C)C3=CC=CC=C3S(=O)(=O)C |
GSK2801是BAZ2家族含溴结构域蛋白的强效抑制剂。
Targets
BAZ2B | BAZ2A | |||
136 nM(Kd) | 257 nM(Kd) |
In vitro (25°C) | DMSO | Warmed: 67 mg/mL (180.37 mM) | |
Water | Insoluble | ||
Ethanol | Warmed: 6 mg/mL (16.15 mM) | ||
In vivo | 0.5% CMC+1% Tween 80 | 28 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 26.92 mL | 134.58 mL | 269.15 mL |
0.5 mM | 5.38 mL | 26.92 mL | 53.83 mL |
1 mM | 2.69 mL | 13.46 mL | 26.92 mL |
5 mM | 0.54 mL | 2.69 mL | 5.38 mL |
*The above data is based on the productmolecular weight 371.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.