TRV130 (Oliceridine)
Catalog No. A14337
TRV130 (Oliceridine)引发强大的G蛋白信号传导，其功效和功效与吗啡相似，但Δε-arrestin2募集和受体内化作用远少于吗啡。
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| Catalog Num | A14337 |
|---|---|
| M. Wt | 423.01 |
| Formula | C22H31ClN2O2S |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1401028-24-7 |
| Synonyms | TRV 130, TRV-130 |
| SMILES | COC1=C(SC=C1)CNCC[C@]2(CCOC3(C2)CCCC3)C4=CC=CC=N4 |
TRV130 (Oliceridine)引发强大的G蛋白信号传导，其功效和功效与吗啡相似，但Δε-arrestin2募集和受体内化作用远少于吗啡。
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.64 mL | 118.2 mL | 236.4 mL |
| 0.5 mM | 4.73 mL | 23.64 mL | 47.28 mL |
| 1 mM | 2.36 mL | 11.82 mL | 23.64 mL |
| 5 mM | 0.47 mL | 2.36 mL | 4.73 mL |
*The above data is based on the productmolecular weight 423.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
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