BQ-123

Catalog No. A15912

BQ-123是一种选择性内皮素A受体(ETA)拮抗剂,IC50为7.3 nM。
Catalog Num A15912
M. Wt 610.7
Formula C31H42N6O7
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 136553-81-6
Synonyms BQ123, BQ 123
SMILES O=C(O)C[C@H]1NC([C@@H](CC2=CNC3=C2C=CC=C3)NC([C@H](CC(C)C)NC([C@@H](C(C)C)NC([C@@](CCC4)([H])N4C1=O)=O)=O)=O)=O
BQ-123是一种选择性内皮素A受体(ETA)拮抗剂,IC50为7.3 nM。
Targets
Endothelin A receptor
7.3 nM
In vitro DMSO Warmed: 87 mg/mL (142.45 mM)
Water Insoluble
Ethanol Warmed: 13 mg/mL (21.29 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.37 mL 81.87 mL 163.75 mL
0.5 mM 3.27 mL 16.37 mL 32.75 mL
1 mM 1.64 mL 8.19 mL 16.37 mL
5 mM 0.33 mL 1.64 mL 3.27 mL

*The above data is based on the productmolecular weight 610.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.