Cyclo (RGDyK) trifluoroacetate

Catalog No. A15918

Cyclo (RGDyK) trifluoroacetate是一种有效的选择性αVbeta3整联蛋白抑制剂，IC50为20 nM。

Technical details

Catalog Num	A15918
M. Wt	847.72
Formula	C31H43F6N9O12
Purity	>98%
Storage	at -20°C 3 years Powder
CAS No.	250612-42-1
Synonyms
SMILES	NCCCC[C@@]1([H])/C(O)=N/[C@@](/C(O)=N/C/C(O)=N/[C@@](/C(O)=N/[C@](/C(O)=N/1)([H])CC2=CC=C(O)C=C2)([H])CC(O)=O)([H])CCCNC(N)=N.FC(F)(F)C(O)=O.FC(F)(F)C(O)=O

Biological Activity

Cyclo (RGDyK) trifluoroacetate是一种有效的选择性αVbeta3整联蛋白抑制剂，IC50为20 nM。

Targets

αVβ3 integrin
20 nM

Solubility *

In vitro	DMSO	97 mg/mL (114.42 mM)
	Water	97 mg/mL (114.42 mM)
	Ethanol	19 mg/mL (22.41 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	11.8 mL	58.98 mL	117.96 mL
0.5 mM	2.36 mL	11.8 mL	23.59 mL
1 mM	1.18 mL	5.9 mL	11.8 mL
5 mM	0.24 mL	1.18 mL	2.36 mL

*The above data is based on the productmolecular weight 847.72. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.