Glucocorticoid receptors

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  1. Mapracorat

    Catalog No. A21953
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    glucocorticoid receptor agonist
    Mapracorat is a novel non-steroidal selective glucocorticoid receptor agonist. 了解更多
  2. (S)-Mapracorat

    Catalog No. A21528
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    glucocorticoid receptor agonist
    (S)-Mapracorat is a selective and less active glucocorticoid receptor agonist. 了解更多
  3. Dagrocorat

    Catalog No. A21312
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    glucocorticoid receptor agonist
    Dagrocorat (PF-00251802) is a novel and dissociated glucocorticoid receptor agonist. 了解更多
  4. Fosdagrocorat

    Catalog No. A21303
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    dissociated glucocorticoid receptor agonist
    Fosdagrocorat (PF-04171327) is a dissociated glucocorticoid receptor agonist. 了解更多
  5. Beclometasone dipropionate

    Catalog No. A17254
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    glucocorticoid agonist
    Beclometasone dipropionate is a potent glucocorticoid agonist; it is a prodrug of the free form, beclometasone. 了解更多
  6. Dexamethasone acetate

    Catalog No. A16494
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    glucocorticoid receptor agonist
    Dexamethasone acetate (Dexamethasone 21-acetate) is a glucocorticoid receptor agonist. 了解更多
  7. Glucocorticoid receptor agonist

    Catalog No. A11431
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    Glucocorticoid receptor agonist
    Glucocorticoid receptor agonist is a potent Glucocorticoid receptor agonist. 了解更多
  8. Betamethasone acibutate

    Catalog No. A18697
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    glucocorticoid
    Betamethasone acibutate, derives from Betamethasone, is an acetate ester. Betamethasone acibutate is a glucocorticoid. 了解更多
  9. AZD2906

    Catalog No. A18936
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    glucocorticoid receptor agonist
    AZD2906 is a selective glucocorticoid receptor (GR) agonist, increases micronucleated immature erythrocytes in the bone marrow of rats. AZD2906 shows IC50s of 2.2, 0.3, 41.6 and 7.5 nM at GR in human, rat PBMC and human, rat whole blood, respectively. 了解更多
  10. Fluorometholone

    Catalog No. A17651
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    glucocorticoid
    Fluorometholone is a glucocorticoid employed, usually as eye drops, in the treatment of allergic and inflammatory conditions of the eye. It has also been used topically in the treatment of various skin disorders. 了解更多
  11. AZD5423

    Catalog No. A13249
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    nonsteroidal glucocorticoid receptor 激动剂
    AZD5423是新型的非甾体类糖皮质激素受体激动剂。 了解更多
  12. RU43044

    Catalog No. A14340
    Glucocorticoid receptor 拮抗剂
    RU43044在骨肉瘤细胞而非人乳腺癌细胞中发挥显着的激动剂活性并激活MMTV-Luc转录。 了解更多
  13. GW-870086

    Catalog No. A18343
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    Glucocorticoid receptor agonist
    GW-870086 is a potent anti-inflammatory agent, acting as a glucocorticoid receptor agonist, with a pIC50 of 10.1 in A549 cells expressing NF-κB. 了解更多
  14. Fluticasone propionate

    Catalog No. A11860
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    Fluticasone propionate是一种高亲和力的选择性糖皮质激素受体激动剂(Kd = 0.5 nM)。 了解更多
  15. Beclometasone

    Catalog No. A18177
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    glucocorticoid receptor agonist
    Beclometasone, also known as Beclomethasone, is an anti-inflammatory, synthetic glucocorticoid. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. 了解更多
  16. AZD9567

    Catalog No. A18850
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    selective glucocorticoid receptor modulator
    AZD9567 is a potent, oral active, non-steroidal and selective glucocorticoid receptor modulator (SGRM), with an IC50 of 3.8 nM. 了解更多
  17. OP-3633

    Catalog No. A18468
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    Glucocorticoid Receptor Antagonist
    OP-3633 is a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (IC50 = 29 nM). 了解更多
  18. Prednisone (Adasone)

    Catalog No. A10752
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    Glucocorticoid Receptor 激动剂
    Prednisone (Adasone)可降低粘膜TNF-a的产生,肠道通透性和NF-kB表达水平。 了解更多
  19. Methylprednisolone

    Catalog No. A10582
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    Methylprednisolone是一种凋亡诱导剂,并且在体外也能抑制人小细胞肺癌细胞的生长。 了解更多
  20. Meprednisone (Betapar)

    Catalog No. A10567
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    Meprednisone是糖皮质激素和泼尼松的甲基化衍生物。 了解更多
  21. Hydrocortisone(Cortisol)

    Catalog No. A10457
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    Hydrocortisone是肾上腺产生的类固醇激素或糖皮质激素。 了解更多
  22. Deflazacort

    Catalog No. A10294
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    Deflazacort是一种糖皮质激素,用作抗炎和免疫抑制剂。 了解更多
  23. Prednisolone acetate (Omnipred)

    Catalog No. A11687
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    Prednisolone是合成的糖皮质激素,是皮质醇的衍生物,用于治疗各种炎症和自身免疫性疾病。 了解更多
  24. Budesonide

    Catalog No. A10166
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    Budesonide是一种糖皮质激素类固醇,可用于治疗哮喘,非感染性鼻炎 了解更多
  25. Betamethasone valerate (Betnovate, Celestone)

    Catalog No. A10131
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    Betamethasone valerate是一种有效的糖皮质激素类固醇,具有抗炎和免疫抑制作用 了解更多
  26. Betamethasone dipropionate

    Catalog No. A10130
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    Glucocorticoid Receptor 激动剂
    Betamethasone Dipropionate是糖皮质激素类固醇,具有抗炎和免疫抑制特性。 了解更多

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