RS-127445

目录号: A11165

5-HT2B receptor 拮抗剂

RS-127445

RS-127445 Chemical Structure

CAS NO. 199864-87-4

RS-127445是5-羟色胺5-HT2B受体的有效和选择性拮抗剂,相对于密切相关的5-HT2A和5-HT2C受体具有约1000倍的选择性。

库存: 现货

规格 价格 数量
5 mg
¥ 400.00
10 mg
¥ 700.00
50 mg
¥ 2,000.00
100 mg
¥ 3,200.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

产品详情

RS-127445是5-羟色胺5-HT2B受体的有效和选择性拮抗剂,相对于密切相关的5-HT2A和5-HT2C受体具有约1000倍的选择性。
靶点信息
5-HT2B 5-HT2B
10.4(pIC50)9.5(pKi)
In vitro DMSO 54 mg/mL (191.94 mM)
Water Insoluble
Ethanol 8 mg/mL (28.43 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 35.55 mL 177.73 mL 355.45 mL
0.5 mM 7.11 mL 35.55 mL 71.09 mL
1 mM 3.55 mL 17.77 mL 35.55 mL
5 mM 0.71 mL 3.55 mL 7.11 mL

*The above data is based on the productmolecular weight 281.33. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11165
作用机制 Antagonist (拮抗剂)
M. Wt 281.33
Formula C17H16FN3
Purity >99%
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

CAS No. 199864-87-4
Synonyms RS127445, MT 500, RS127,445
SMILES CC(C)C1=NC(=NC(=C1)C2=CC=C(C3=CC=CC=C32)F)N.Cl

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