RS-127445

目录号: A11165

5-HT2B receptor antagonist

RS-127445

RS-127445 Chemical Structure

CAS NO. 199864-87-4

RS-127445 is a potent and selective antagonist at the serotonin 5-HT2B receptor, with around 1000x selectivity over the closely related 5-HT2A and 5-HT2C receptors.

库存: 现货

规格 价格 数量
5 mg
¥ 400.00
10 mg
¥ 700.00
50 mg
¥ 2,000.00
100 mg
¥ 3,200.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

RS-127445 is a potent and selective antagonist at the serotonin 5-HT2B receptor, with around 1000x selectivity over the closely related 5-HT2A and 5-HT2C receptors.

Targets
5-HT2B 5-HT2B
10.4(pIC50)9.5(pKi)
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 35.55 mL 177.73 mL 355.45 mL
0.5 mM 7.11 mL 35.55 mL 71.09 mL
1 mM 3.55 mL 17.77 mL 35.55 mL
5 mM 0.71 mL 3.55 mL 7.11 mL

*The above data is based on the productmolecular weight 281.33. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

目录号 A11165
MECHANISM OF ACTION Antagonist
M. Wt 281.33
Formula C17H16FN3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 199864-87-4
Synonyms RS127445, MT 500, RS127,445
SMILES CC(C)C1=NC(=NC(=C1)C2=CC=C(C3=CC=CC=C32)F)N.Cl

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