GSK1292263

Catalog No. A10439

GSK-1292263是一种新型GPR119激动剂。

Product Citations

Inoue A, .et al. Illuminating G-Protein-Coupling Selectivity of GPCRs, Cell, 2019, Jun 13;177(7):1933-1947 PMID: 31160049

Technical details

Catalog Num	A10439
M. Wt	456.6
Formula	C23H28N4O4S
Purity	>98%
Storage	at -20°C 3 years Powder
CAS No.	1032823-75-8
Synonyms	GSK-1292263
SMILES	CC(C)C1=NOC(=N1)N2CCC(CC2)COC3=CN=C(C=C3)C4=CC=C(C=C4)S(=O)(=O)C

Biological Activity

GSK-1292263是一种新型GPR119激动剂。

Targets

GPR119

Solubility *

In vitro (25°C)	DMSO	29 mg/mL (63.51 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	30% propylene glycol, 5% Tween 80, 65% D5W	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.9 mL	109.51 mL	219.01 mL
0.5 mM	4.38 mL	21.9 mL	43.8 mL
1 mM	2.19 mL	10.95 mL	21.9 mL
5 mM	0.44 mL	2.19 mL	4.38 mL

*The above data is based on the productmolecular weight 456.6. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.