Ketanserin (Vulketan Gel)
Catalog No. A10497
Ketanserin (Vulketan Gel)是大鼠和人5-HT2A血清素受体拮抗剂,Ki为2.5 nM。
Catalog Num | A10497 |
---|---|
M. Wt | 395.43 |
Formula | C22H22FN3O3 |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 74050-98-9 |
Synonyms | R 41468, Vulketan Gel |
SMILES | C1CN(CCC1C(=O)C2=CC=C(C=C2)F)CCN3C(=O)C4=CC=CC=C4NC3=O |
Ketanserin (Vulketan Gel)是大鼠和人5-HT2A血清素受体拮抗剂,Ki为2.5 nM。
Targets
5-HT2A | 5-HT2C (Rat) | 5-HT2C (Human) | ||
2.5 nM(Ki) | 50 nM(Ki) | 100 nM(Ki) |
In vitro (25°C) | DMSO | 2 mg/mL (5.05 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
In vivo | 4% DMSO+40% PEG 300+4% Tween 80+ddH2O | 1 mg/mL | |
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 25.29 mL | 126.44 mL | 252.89 mL |
0.5 mM | 5.06 mL | 25.29 mL | 50.58 mL |
1 mM | 2.53 mL | 12.64 mL | 25.29 mL |
5 mM | 0.51 mL | 2.53 mL | 5.06 mL |
*The above data is based on the productmolecular weight 395.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.