Rupatadine Fumarate
Catalog No. A12356
Rupatadine Fumarate是PAFR和组胺(H1)受体的抑制剂,Ki分别为550和102 nM。
Catalog Num | A12356 |
---|---|
M. Wt | 532.03 |
Formula | C26H26ClN3.C4H4O4 |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 182349-12-8 |
Synonyms | |
SMILES | CC1=CC(=CN=C1)CN2CCC(=C3C4=C(CCC5=C3N=CC=C5)C=C(C=C4)Cl)CC2.C(=C/C(=O)O)\C(=O)O |
Rupatadine Fumarate是PAFR和组胺(H1)受体的抑制剂,Ki分别为550和102 nM。
Targets
Histamine H1 receptor | PAFR | |||
102 nM(Ki) | 550 nM(Ki) |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 18.8 mL | 93.98 mL | 187.96 mL |
0.5 mM | 3.76 mL | 18.8 mL | 37.59 mL |
1 mM | 1.88 mL | 9.4 mL | 18.8 mL |
5 mM | 0.38 mL | 1.88 mL | 3.76 mL |
*The above data is based on the productmolecular weight 532.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.