SR 144528
Catalog No. A12376
SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。
- Ming Tang, .et al. Celastrol alleviates renal fibrosis by upregulating cannabinoid receptor 2 expression, Cell Death Dis, 2018, Jun; 9(6): 601 PMID: 29789558
| Catalog Num | A12376 |
|---|---|
| M. Wt | 476.05 |
| Formula | C29H34ClN3O |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 192703-06-3 |
| Synonyms | SR144528, SR-144528 |
| SMILES | CC1=CC=C(C=C1)CN2C(=CC(=N2)C(=O)N[C@H]3[C@]4(CC[C@H](C4)C3(C)C)C)C5=CC(=C(C=C5)Cl)C |
SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.01 mL | 105.03 mL | 210.06 mL |
| 0.5 mM | 4.2 mL | 21.01 mL | 42.01 mL |
| 1 mM | 2.1 mL | 10.5 mL | 21.01 mL |
| 5 mM | 0.42 mL | 2.1 mL | 4.2 mL |
*The above data is based on the productmolecular weight 476.05. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Contact information
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
ADOOQ 产品质量保证
We promise all products to perform as described.