CPI 0610

Catalog No. A16076

CPI 0610是Bromodomain和Extra-Terminal（BET）蛋白家族的小分子抑制剂，具有潜在的抗肿瘤活性。

Technical details

Catalog Num	A16076
M. Wt	365.82
Formula	C20H16ClN3O2
Purity	>98%
Storage	at -20°C 3 years Powder
CAS No.	1380087-89-7
Synonyms	CPI0610, CPI-0610
SMILES	O=C(N)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C3=CC=CC=C3C4=C1ON=C4C

Biological Activity

CPI 0610是Bromodomain和Extra-Terminal（BET）蛋白家族的小分子抑制剂，具有潜在的抗肿瘤活性。

Targets

BRD4-BD1	MYC
39 nM	180 nM(EC50)

Solubility *

In vitro	DMSO	70 mg/mL (191.35 mM)
	Water	Insoluble
	Ethanol	12 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	27.34 mL	136.68 mL	273.36 mL
0.5 mM	5.47 mL	27.34 mL	54.67 mL
1 mM	2.73 mL	13.67 mL	27.34 mL
5 mM	0.55 mL	2.73 mL	5.47 mL

*The above data is based on the productmolecular weight 365.82. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.