ERK5-IN-1
Catalog No. A16232
ERK5-IN-1表现出对ERK5的有效抑制,其细胞EC50值为0.19 uM,酶促IC50值为0.087 uM,LRRK2 [G2019S]具有酶促IC50值为0.026uM。
Catalog Num | A16232 |
---|---|
M. Wt | 459.54 |
Formula | C25H29N7O2 |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1234479-76-5 |
Synonyms | ERK5 IN 1, ERK5IN1 |
SMILES | O=C1N(C)C2=CN=C(NC3=CC=C(N4CCN(C)CC4)C=C3OC)N=C2N(C)C5=CC=CC=C15 |
ERK5-IN-1表现出对ERK5的有效抑制,其细胞EC50值为0.19 uM,酶促IC50值为0.087 uM,LRRK2 [G2019S]具有酶促IC50值为0.026uM。
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 21.76 mL | 108.8 mL | 217.61 mL |
0.5 mM | 4.35 mL | 21.76 mL | 43.52 mL |
1 mM | 2.18 mL | 10.88 mL | 21.76 mL |
5 mM | 0.44 mL | 2.18 mL | 4.35 mL |
*The above data is based on the productmolecular weight 459.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.