TGR-1202 hydrochloride (Umbralisib HCl)
Catalog No. A16278
TGR-1202 hydrochloride是一种口服的下一代PI3Kδ抑制剂，在基于酶和细胞的测定中抑制PI3Kδ活性，IC50和EC50值分别为22.2和24.3 nM。
| Catalog Num | A16278 |
|---|---|
| M. Wt | 608.01 |
| Formula | C31H25ClF3N5O3 |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1532533-78-0 |
| Synonyms | RP5264 hydrochloride, TGR1202 hydrochloride, TGR 1202 hydrochloride, RP-5264 hydrochloride, RP 5264 hydrochloride |
| SMILES | O=C1C(C2=CC=CC(F)=C2)=C([C@@H](N3N=C(C4=CC=C(OC(C)C)C(F)=C4)C5=C(N)N=CN=C53)C)OC6=CC=C(F)C=C16.[H]Cl |
TGR-1202 hydrochloride是一种口服的下一代PI3Kδ抑制剂，在基于酶和细胞的测定中抑制PI3Kδ活性，IC50和EC50值分别为22.2和24.3 nM。
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 16.45 mL | 82.24 mL | 164.47 mL |
| 0.5 mM | 3.29 mL | 16.45 mL | 32.89 mL |
| 1 mM | 1.64 mL | 8.22 mL | 16.45 mL |
| 5 mM | 0.33 mL | 1.64 mL | 3.29 mL |
*The above data is based on the productmolecular weight 608.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Contact information
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
ADOOQ 产品质量保证
We promise all products to perform as described.