Flupirtine maleate

Catalog No. A10251

Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。

Technical details

Catalog Num	A10251
M. Wt	420.4
Formula	C15H17FN4O2.C4H4O4
Purity	>98%
Storage	at -20°C 3 years Powder
CAS No.	75507-68-5
Synonyms	D 9998
SMILES	CCOC(=O)NC1=C(N=C(C=C1)NCC2=CC=C(C=C2)F)N.C(=C\C(=O)O)\C(=O)O

Biological Activity

Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。

Targets

NMDA receptor	Potassium channel

Solubility *

In vitro (25°C)	DMSO	76 mg/mL (180.78 mM)
	Water	Insoluble
	Ethanol	Warmed: 2 mg/mL (4.75 mM)
In vivo	30% propylene glycol, 5% Tween 80, 65% D5W	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	23.79 mL	118.93 mL	237.87 mL
0.5 mM	4.76 mL	23.79 mL	47.57 mL
1 mM	2.38 mL	11.89 mL	23.79 mL
5 mM	0.48 mL	2.38 mL	4.76 mL

*The above data is based on the productmolecular weight 420.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.