RGFP966

Catalog No. A13218

RGFP966是一种HDAC3抑制剂,IC50为0.08μM,与其他HDAC相比,具有> 200倍的选择性。
Catalog Num A13218
M. Wt 362.4
Formula C21H19FN4O
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1357389-11-7
Synonyms RGFP-966, RGFP 966
SMILES C1=CC=C(C=C1)/C=C/CN2C=C(C=N2)/C=C/C(=O)NC3=C(C=C(C=C3)F)N
RGFP966是一种HDAC3抑制剂,IC50为0.08μM,与其他HDAC相比,具有> 200倍的选择性。
In vitro (25°C) DMSO 70 mg/mL (193.15 mM)
Water Insoluble
Ethanol Insoluble
In vivo 5%DMSO+40%PEG300+10%Tween80+45%ddH2O 6.1 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.59 mL 137.97 mL 275.94 mL
0.5 mM 5.52 mL 27.59 mL 55.19 mL
1 mM 2.76 mL 13.8 mL 27.59 mL
5 mM 0.55 mL 2.76 mL 5.52 mL

*The above data is based on the productmolecular weight 362.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.