Eprosartan mesylate

Catalog No. A13747

Eprosartan mesylate是一种竞争性的AT1受体拮抗剂,IC50值为1.4-3.9 nM,消除半衰期为5至7小时。
Catalog Num A13747
M. Wt 520.6
Formula C23H24N2O4S ? CH3SO3H
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 144143-96-4
Synonyms SKF 108566J
SMILES CCCCC1=NC=C(N1CC2=CC=C(C=C2)C(=O)O)/C=C(\CC3=CC=CS3)/C(=O)O.CS(=O)(=O)O
Eprosartan mesylate是一种竞争性的AT1受体拮抗剂,IC50值为1.4-3.9 nM,消除半衰期为5至7小时。
In vitro DMSO 97 mg/mL (186.31 mM)
Water Insoluble
Ethanol 4 mg/mL (7.68 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.21 mL 96.04 mL 192.09 mL
0.5 mM 3.84 mL 19.21 mL 38.42 mL
1 mM 1.92 mL 9.6 mL 19.21 mL
5 mM 0.38 mL 1.92 mL 3.84 mL

*The above data is based on the productmolecular weight 520.6. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.