Atipamezole HCl

Catalog No. A13902

Atipamezole hydrochloride是一种选择性α2肾上腺素受体拮抗剂（α2A、α2B、α2C、α1A和α1B受体的Ki值分别为1.1、1.0、0.89、1300和6500nm）。已经被证明是大脑的渗透剂。

Technical details

Catalog Num	A13902
M. Wt	248.8
Formula	C14H16N2.HCl
Purity	>98%
Storage	at -20°C 3 years Powder
CAS No.	104075-48-1
Synonyms	Antisedan
SMILES	CCC1(CC2=CC=CC=C2C1)C3=CN=CN3.Cl

Biological Activity

Targets

α2 adrenergic receptor

Solubility *

In vitro	DMSO	12 mg/mL (48.24 mM)
	Water	21 mg/mL (84.42 mM)
	Ethanol	48 mg/mL (192.96 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	40.19 mL	200.96 mL	401.93 mL
0.5 mM	8.04 mL	40.19 mL	80.39 mL
1 mM	4.02 mL	20.1 mL	40.19 mL
5 mM	0.8 mL	4.02 mL	8.04 mL

*The above data is based on the productmolecular weight 248.8. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.