Talabostat
Catalog No. A14079
Talabostat (Val-boroPro; PT100) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 < 4 nM; Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM).
Catalog Num | A14079 |
---|---|
M. Wt | 214.07 |
Formula | C9H19BN2O3 |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 149682-77-9 |
Synonyms | Val-boroPro; PT100 |
SMILES | CC(C)[C@H](N)C(N1[C@H](B(O)O)CCC1)=O |
Talabostat (Val-boroPro; PT100) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 < 4 nM; Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM).
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 46.71 mL | 233.57 mL | 467.14 mL |
0.5 mM | 9.34 mL | 46.71 mL | 93.43 mL |
1 mM | 4.67 mL | 23.36 mL | 46.71 mL |
5 mM | 0.93 mL | 4.67 mL | 9.34 mL |
*The above data is based on the productmolecular weight 214.07. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.