Talabostat

Catalog No. A14079

Talabostat (Val-boroPro; PT100) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 < 4 nM; Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM).
Catalog Num A14079
M. Wt 214.07
Formula C9H19BN2O3
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 149682-77-9
Synonyms Val-boroPro; PT100
SMILES CC(C)[C@H](N)C(N1[C@H](B(O)O)CCC1)=O
Talabostat (Val-boroPro; PT100) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 < 4 nM; Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 46.71 mL 233.57 mL 467.14 mL
0.5 mM 9.34 mL 46.71 mL 93.43 mL
1 mM 4.67 mL 23.36 mL 46.71 mL
5 mM 0.93 mL 4.67 mL 9.34 mL

*The above data is based on the productmolecular weight 214.07. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.