GSK-2193874
Catalog No. A14201
GSK2193874被确定为选择性的口服活性TRPV4阻滞剂，可通过重组TRPV4通道和天然内皮TRPV4电流抑制Ca(2+)流入。
| Catalog Num | A14201 |
|---|---|
| M. Wt | 691.62 |
| Formula | C37H38BrF3N4O |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 1336960-13-4 |
| Synonyms | GSK 2193874, GSK2193874 |
| SMILES | C1CCN(CC1)C2CCN(CC2)CC3=C(N=C4C=C(C=CC4=C3C(=O)NC5(CC5)C6=CC=CC=C6)Br)C7=CC(=CC=C7)C(F)(F)F |
GSK2193874被确定为选择性的口服活性TRPV4阻滞剂，可通过重组TRPV4通道和天然内皮TRPV4电流抑制Ca(2+)流入。
| In vitro | DMSO | 95 mg/mL (137.35 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 48 mg/mL (69.4 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 14.46 mL | 72.29 mL | 144.59 mL |
| 0.5 mM | 2.89 mL | 14.46 mL | 28.92 mL |
| 1 mM | 1.45 mL | 7.23 mL | 14.46 mL |
| 5 mM | 0.29 mL | 1.45 mL | 2.89 mL |
*The above data is based on the productmolecular weight 691.62. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Contact information
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
ADOOQ 产品质量保证
We promise all products to perform as described.