SB-408124 HCl
Catalog No. A15231
SB408124 Hydrochloride是OX1受体的非肽拮抗剂,全细胞和膜的Ki分别为57 nM和27 nM。表现出比OX2受体高50倍的选择性。
Catalog Num | A15231 |
---|---|
M. Wt | 392.83 |
Formula | C19H19ClF2N4O |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1431697-90-3 |
Synonyms | SB 408124 Hydrochloride, SB408124 Hydrochloride |
SMILES | CC1=NC2=C(C=C(C=C2C(=C1)NC(=O)NC3=CC=C(C=C3)N(C)C)F)F.Cl |
SB408124 Hydrochloride是OX1受体的非肽拮抗剂,全细胞和膜的Ki分别为57 nM和27 nM。表现出比OX2受体高50倍的选择性。
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 25.46 mL | 127.28 mL | 254.56 mL |
0.5 mM | 5.09 mL | 25.46 mL | 50.91 mL |
1 mM | 2.55 mL | 12.73 mL | 25.46 mL |
5 mM | 0.51 mL | 2.55 mL | 5.09 mL |
*The above data is based on the productmolecular weight 392.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.