CRT-0066101

Catalog No. A16318

CRT-0066101是有效，选择性的蛋白激酶D（PKD）抑制剂；抑制所有PKD同工型（PKD1，PKD3和PKD2的IC50值分别为1、2和2.5 nM）。

Technical details

Catalog Num	A16318
M. Wt	411.33
Formula	C18H22N6O.2HCl
Purity	>98%
Storage	at -20°C 3 years Powder
CAS No.	1883545-60-5
Synonyms	CRT 0066101, CRT0066101
SMILES	Cl.Cl.Cn1cc(cn1)c3cc(c2nc(NC[C@H](N)CC)ccn2)c(O)cc3

Biological Activity

CRT-0066101是有效，选择性的蛋白激酶D（PKD）抑制剂；抑制所有PKD同工型（PKD1，PKD3和PKD2的IC50值分别为1、2和2.5 nM）。

Solubility *

In vitro	DMSO	Warmed: 25 mg/mL (60.77 mM)
	Water	80 mg/mL (194.49 mM)
	Ethanol	Warmed: 2 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	24.31 mL	121.56 mL	243.11 mL
0.5 mM	4.86 mL	24.31 mL	48.62 mL
1 mM	2.43 mL	12.16 mL	24.31 mL
5 mM	0.49 mL	2.43 mL	4.86 mL

*The above data is based on the productmolecular weight 411.33. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Adooq Bioscience

CRT-0066101

Technical details

Biological Activity

Solubility *

Preparing Stock Solutions