ASTX-660

Catalog No. A16996

ASTX660是X染色体连锁的凋亡蛋白抑制剂（XIAP）和细胞IAP 1（cIAP1）的口服生物利用型非拟肽拮抗剂，具有潜在的抗肿瘤和促凋亡活性。1799328-86-1 (free base) 1799328-50-9 (HCl) 1799328-90-7 (mesylate) 1799328-88-3 (sulfate)

Technical details

Catalog Num	A16996
M. Wt	539.69
Formula	C30H42FN5O3
Purity	>98%
Storage	at -20°C 3 years Powder
CAS No.	1799328-86-1
Synonyms	ASTX660, ASTX 660
SMILES	OCC1=NC2=C(N(CC2(C)C)C(CN3[C@@H](CN4[C@H](C)COCC4)CN[C@H](C)C3)=O)C=C1CC5=CC=C(F)C=C5

Solubility *

In vitro	DMSO	93 mg/mL (172.32 mM)
	Water	Insoluble
	Ethanol	93 mg/mL (172.32 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	18.53 mL	92.65 mL	185.29 mL
0.5 mM	3.71 mL	18.53 mL	37.06 mL
1 mM	1.85 mL	9.26 mL	18.53 mL
5 mM	0.37 mL	1.85 mL	3.71 mL

*The above data is based on the productmolecular weight 539.69. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Adooq Bioscience

ASTX-660

Technical details

Biological Activity

Solubility *

Preparing Stock Solutions