BETd-246

Catalog No. A18913

BETd-246 is a second-generation BET bromodomain (BRD) inhibitor, exhibiting superior selectivity, potency and antitumor activity.
Catalog Num A18913
M. Wt 946.03
Formula C48H55N11O10
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2140289-17-2
Synonyms BETd-246; BETd 246; BETd246
SMILES O=C(C1=NC(NC2=CC(C3CC3)=NN2CC)=C4C(NC5=C4C=C(OC)C(C6=C(C)ON=C6C)=C5)=N1)NCCCOCCOCCOCCCNC7=CC=CC(C(N8C(CC9)C(NC9=O)=O)=O)=C7C8=O
BETd-246 is a second-generation BET bromodomain (BRD) inhibitor, exhibiting superior selectivity, potency and antitumor activity.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 10.57 mL 52.85 mL 105.7 mL
0.5 mM 2.11 mL 10.57 mL 21.14 mL
1 mM 1.06 mL 5.29 mL 10.57 mL
5 mM 0.21 mL 1.06 mL 2.11 mL

*The above data is based on the productmolecular weight 946.03. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.