PROTAC BET Degrader-1

Catalog No. A20016

PROTAC BET Degrader-1 is a potent BET degrader based on PROTAC, decreasing BRD2, BRD3, and BRD4 protein levels at low concentration.
Catalog Num A20016
M. Wt 871.9
Formula C44H45N11O9
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2093386-22-0
Synonyms
SMILES CCN1C(NC2=C3C4=CC(OC)=C(C(C(C)=NO5)=C5C)C=C4NC3=NC(C(NCCCCNC(COC6=C(C(N7C(CCC8=O)C(N8)=O)=O)C(C7=O)=CC=C6)=O)=O)=N2)=CC(C9CC9)=N1
PROTAC BET Degrader-1 is a potent BET degrader based on PROTAC, decreasing BRD2, BRD3, and BRD4 protein levels at low concentration.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 11.47 mL 57.35 mL 114.69 mL
0.5 mM 2.29 mL 11.47 mL 22.94 mL
1 mM 1.15 mL 5.73 mL 11.47 mL
5 mM 0.23 mL 1.15 mL 2.29 mL

*The above data is based on the productmolecular weight 871.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.