GLP-1R Antagonist 1
Catalog No. A20679
GLP-1R Antagonist 1 (compound 5d) is an orally active, CNS penetrant and non-competitive antagonist of glucagon-like peptide 1 receptor (GLP-1R), with an IC50 of 650 nM.
| Catalog Num | A20679 |
|---|---|
| M. Wt | 440.73 |
| Formula | C16H11ClF6N4O2 |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 488097-06-9 |
| Synonyms | |
| SMILES | O=C1C2=C(NC(C3=CC=C(Cl)C=C3)=NC2(C(F)(F)F)C(F)(F)F)N(C)C(N1C)=O |
GLP-1R Antagonist 1 (compound 5d) is an orally active, CNS penetrant and non-competitive antagonist of glucagon-like peptide 1 receptor (GLP-1R), with an IC50 of 650 nM.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 22.69 mL | 113.45 mL | 226.9 mL |
| 0.5 mM | 4.54 mL | 22.69 mL | 45.38 mL |
| 1 mM | 2.27 mL | 11.34 mL | 22.69 mL |
| 5 mM | 0.45 mL | 2.27 mL | 4.54 mL |
*The above data is based on the productmolecular weight 440.73. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
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