GSK180736A

Catalog No. A20736

GSK180736A is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 μM.
Catalog Num A20736
M. Wt 365.36
Formula C19H16FN5O2
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 817194-38-0
Synonyms GSK-180736A; GSK 180736A
SMILES CC(N1)=C(C(NC2=CC=C(NN=C3)C3=C2)=O)C(C4=CC=C(F)C=C4)NC1=O
GSK180736A is a G protein-coupled receptor kinase 2 (GRK2) inhibitor with an IC50 of 0.77 μM.
In vitro DMSO Warmed: 66 mg/mL (180.64 mM)
Water Insoluble
Ethanol Warmed: 3 mg/mL (8.21 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.37 mL 136.85 mL 273.7 mL
0.5 mM 5.47 mL 27.37 mL 54.74 mL
1 mM 2.74 mL 13.69 mL 27.37 mL
5 mM 0.55 mL 2.74 mL 5.47 mL

*The above data is based on the productmolecular weight 365.36. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.