(R)-Elagolix

Catalog No. A21184

Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM).
Catalog Num A21184
M. Wt 631.59
Formula C32H30F5N3O5
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 834153-87-6
Synonyms NBI-56418, NBI56418, NBI 56418
SMILES FC1=C(C2=C(C)N(CC3=C(C(F)(F)F)C=CC=C3F)C(N(C[C@](C4=CC=CC=C4)([H])NCCCC(O)=O)C2=O)=O)C=CC=C1OC
Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 15.83 mL 79.17 mL 158.33 mL
0.5 mM 3.17 mL 15.83 mL 31.67 mL
1 mM 1.58 mL 7.92 mL 15.83 mL
5 mM 0.32 mL 1.58 mL 3.17 mL

*The above data is based on the productmolecular weight 631.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.