Capsazepine

Catalog No. A21208

Capsazepine is a synthetic analogue of the sensory neurone excitotoxin, and an antagonist of TRPV1 receptor with an IC50 of 562 nM.
Catalog Num A21208
M. Wt 376.9
Formula C19H21ClN2O2S
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 138977-28-3
Synonyms
SMILES S=C(N1CCCC2=CC(O)=C(O)C=C2C1)NCCC3=CC=C(Cl)C=C3
Capsazepine is a synthetic analogue of the sensory neurone excitotoxin, and an antagonist of TRPV1 receptor with an IC50 of 562 nM.
In vitro DMSO 68 mg/mL (180.42 mM)
Water Insoluble
Ethanol 68 mg/mL (180.42 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 26.53 mL 132.66 mL 265.32 mL
0.5 mM 5.31 mL 26.53 mL 53.06 mL
1 mM 2.65 mL 13.27 mL 26.53 mL
5 mM 0.53 mL 2.65 mL 5.31 mL

*The above data is based on the productmolecular weight 376.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.