Teneligliptin hydrobromide hydrate

Catalog No. A21465

Teneligliptin hydrobromide hydrate is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM.
Catalog Num A21465
M. Wt 426.58
Formula C22H30N6OS
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1572583-29-9
Synonyms MP-513 hydrobromide hydrate, MP513, MP 513
SMILES CC1=NN(C2=CC=CC=C2)C(N3CCN([C@]4([H])CN[C@H](C(N5CSCC5)=O)C4)CC3)=C1.CC6=NN(C7=CC=CC=C7)C(N8CCN([C@]9([H])CN[C@H](C(N%10CSCC%10)=O)C9)CC8)=C6.Br.Br.Br.Br.Br.O
Teneligliptin hydrobromide hydrate is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.44 mL 117.21 mL 234.42 mL
0.5 mM 4.69 mL 23.44 mL 46.88 mL
1 mM 2.34 mL 11.72 mL 23.44 mL
5 mM 0.47 mL 2.34 mL 4.69 mL

*The above data is based on the productmolecular weight 426.58. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.