GSK2807 Trifluoroacetate

Catalog No. A21731

GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM.
Catalog Num A21731
M. Wt 566.53
Formula C21H33F3N8O7
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2245255-66-5
Synonyms GSK 2807, GSK-2807
SMILES NC1=C2C(N([C@H]3[C@H](O)[C@H](O)[C@@H](CN(CC[C@H](N)C(O)=O)CCCN(C)C)O3)C=N2)=NC=N1.OC(C(F)(F)F)=O
GSK2807 Trifluoroacetate is a potent, selective and SAM-competitive inhibitor of SMYD3, with a Ki of 14 nM and an IC50 of 130 nM.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.65 mL 88.26 mL 176.51 mL
0.5 mM 3.53 mL 17.65 mL 35.3 mL
1 mM 1.77 mL 8.83 mL 17.65 mL
5 mM 0.35 mL 1.77 mL 3.53 mL

*The above data is based on the productmolecular weight 566.53. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.