GK921

Catalog No. A21785

GK921 is a transglutaminase 2 (TGase) inhibitor with an IC50 of 7.71 μM for human recombinant TGase 2.
Catalog Num A21785
M. Wt 344.41
Formula C21H20N4O
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1025015-40-0
Synonyms GK 921, GK-921
SMILES C12=NC=CC=C1N=C(OCCN3CCCC3)C(C#CC4=CC=CC=C4)=N2
GK921 is a transglutaminase 2 (TGase) inhibitor with an IC50 of 7.71 μM for human recombinant TGase 2.
In vitro DMSO 31 mg/mL (90 mM)
Water
Ethanol
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.04 mL 145.18 mL 290.35 mL
0.5 mM 5.81 mL 29.04 mL 58.07 mL
1 mM 2.9 mL 14.52 mL 29.04 mL
5 mM 0.58 mL 2.9 mL 5.81 mL

*The above data is based on the productmolecular weight 344.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.