(Rac)-VU 6008667

Catalog No. A21939

(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration.
Catalog Num A21939
M. Wt 438.85
Formula C24H17ClF2N2O2
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2092917-63-8
Synonyms VU6008667, VU-6008667
SMILES O=C1N2C(N(C(C3=CC=C(F)C(F)=C3)=O)CC2)(C4=CC=C(Cl)C(C)=C4)C5=C1C=CC=C5
(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.79 mL 113.93 mL 227.87 mL
0.5 mM 4.56 mL 22.79 mL 45.57 mL
1 mM 2.28 mL 11.39 mL 22.79 mL
5 mM 0.46 mL 2.28 mL 4.56 mL

*The above data is based on the productmolecular weight 438.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.