MM-102 TFA

Catalog No. A21941

MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide.
Catalog Num A21941
M. Wt 783.83
Formula C37H50F5N7O6
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1883545-52-5
Synonyms HMTase Inhibitor IX TFA, MM102, MM 102
SMILES O=C(C1(NC([C@@H](NC(C(NC(C(C)C)=O)(CC)CC)=O)CCCNC(N)=N)=O)CCCC1)NC(C2=CC=C(F)C=C2)C3=CC=C(F)C=C3.FC(F)(F)C(O)=O
MM-102 TFA (HMTase Inhibitor IX TFA) is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM with an estimated Ki < 1 nM in WDR5 binding assay, which is >200 times more potent than the ARA peptide.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.76 mL 63.79 mL 127.58 mL
0.5 mM 2.55 mL 12.76 mL 25.52 mL
1 mM 1.28 mL 6.38 mL 12.76 mL
5 mM 0.26 mL 1.28 mL 2.55 mL

*The above data is based on the productmolecular weight 783.83. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.