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5-hydroxymethyl tolterodine (PNU 200577)

5-hydroxymethyl tolterodine (PNU 200577)

Name: 5-hydroxymethyl tolterodine (PNU 200577)
SKU: A11166

目录号: A11166

muscarinic receptor 拮抗剂

5-hydroxymethyl tolterodine (PNU 200577) Chemical Structure

CAS NO. 207679-81-0

5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。

库存：现货

规格	价格	数量
5 mg	￥ 1,600.00
10 mg	￥ 2,800.00
50 mg	￥ 6,800.00
100 mg	￥ 10,500.00
10mM * 1mL in DMSO	￥ 1,680.00

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产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。

靶点信息

mAChR
0.84 nM(Kb)

溶解度 *

In vitro	DMSO	60 mg/mL (175.69 mM)
	Water	Insoluble
	Ethanol	60 mg/mL (175.69 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	29.28 mL	146.42 mL	292.83 mL
0.5 mM	5.86 mL	29.28 mL	58.57 mL
1 mM	2.93 mL	14.64 mL	29.28 mL
5 mM	0.59 mL	2.93 mL	5.86 mL

*The above data is based on the productmolecular weight 341.49. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11166
作用机制	Antagonist (拮抗剂)
M. Wt	341.49
Formula	C22H31NO2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	207679-81-0
Synonyms	(R)-5-Hydroxymethyl tolterodine
SMILES	CC(C)N(CC[C@H](C1=CC=CC=C1)C2=C(C=CC(=C2)CO)O)C(C)C