9-Phenanthrol
目录号: A17570
TRPM4 blocker
选择性TRPM4阻断剂(在HEK293细胞中的IC50 = 20 μM)。对CFTR或TRPM5无影响(分别在0.25 mM和1 mM浓度下)。在小鼠心脏模型中消除由缺氧引起的心律失常。
Discription | Selective TRPM4 blocker (IC50 = 20 μM in HEK293 cells). Exhibits no effect on CFTR or TRPM5 (at 0.25 and 1 mM respectively). Abolishes arrhythmias induced by hypoxia in a mouse heart model. |
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目录号 | A17570 |
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分子式 | C14H10O |
分子量 | 194.23 |
CAS号 | 484-17-3 |
SMILES | C1=CC=C2C(=C1)C=C(C3=CC=CC=C23)O |
其他名称 | phenanthren-9-ol |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2