A-438079 HCl
目录号: A12597
P2X7 receptor 拮抗剂
A-438079 HCl 是一种竞争性 P2X7 受体拮抗剂(pIC50 = 6.9,用于抑制人类重组 P2X7 细胞系中的 Ca2+ 流入)。在其他 P2 受体 上没有活性(IC50 >> 10 uM)。
Discription | A-438079 HCl is a competitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line). Devoid of activity at other P2 receptors (IC50 >> 10 uM). |
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目录号 | A12597 |
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分子式 | C13H10Cl3N5 |
分子量 | 342.608 |
CAS号 | 899507-36-9 |
SMILES | ClC1=CC=CC(C2=NN=NN2CC3=CN=CC=C3)=C1Cl.Cl |
其他名称 | A-438079 , A 438079, A438079, A-438079 HCl |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2