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Citarinostat (ACY-241)

Citarinostat (ACY-241)

Name: Citarinostat (ACY-241)
SKU: A12758

目录号: A12758

HDAC6 抑制剂

Product Citations (1)

Citarinostat (ACY-241) Chemical Structure

CAS NO. 1316215-12-9

ACY-241是HDAC6的新型，选择性和口服抑制剂。对HDAC6和HDAC3的IC50分别为2.6 nM和46 nM。

库存：现货

规格	价格	数量
5 mg	￥ 1,200.00
10 mg	￥ 2,000.00
25 mg	￥ 4,000.00

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生物活性

ACY-241是HDAC6的新型，选择性和口服抑制剂。对HDAC6和HDAC3的IC50分别为2.6 nM和46 nM。

溶解度 *

In vitro	DMSO	39 mg/mL (83.34 mM)
	Water	Insoluble
	Ethanol	87 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.37 mL	106.85 mL	213.7 mL
0.5 mM	4.27 mL	21.37 mL	42.74 mL
1 mM	2.14 mL	10.68 mL	21.37 mL
5 mM	0.43 mL	2.14 mL	4.27 mL

*The above data is based on the productmolecular weight 467.95. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A12758
作用机制	Inhibitor (抑制剂)
M. Wt	467.95
Formula	C24H26ClN5O3
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	1316215-12-9
Synonyms	HDAC-IN-2
SMILES	ClC1=CC=CC=C1N(C2=CC=CC=C2)C3=NC=C(C=N3)C(NCCCCCCC(NO)=O)=O