ADL5859 HCl
目录号: A11072
Opioid Receptor 激动剂
ADL5859 HCl 是一种高效且选择性的 δ 阿片受体激动剂,其 Ki 值为 0.84 nM,ED50 值为 20 nM。
| Discription | ADL5859 HCl is a highly potent and selective δ opioid receptor agonist with Ki value to be 0.84 nM and ED50 value to be 20 nM. | ||
|---|---|---|---|
| Targets |
|
| 目录号 | A11072 |
|---|---|
| 分子式 | C24H28N2O3.HCl |
| 分子量 | 429 |
| CAS号 | 850173-95-4 |
| SMILES | CCN(CC)C(=O)C1=CC=C(C=C1)C2=CC3(CCNCC3)OC4=C2C(=CC=C4)O.Cl |
| 其他名称 | ADL-5859 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
| In vitro (25°C) | DMSO | 76 mg/mL (177.17 mM) | |
| Water | 4 mg/mL (9.32 mM) | ||
| Ethanol | 1 mg/mL (2.33 mM) | ||
| In vivo | 0.5% hydroxyethyl cellulose+0.1% Tween 80 | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.31 mL | 116.55 mL | 233.1 mL |
| 0.5 mM | 4.66 mL | 23.31 mL | 46.62 mL |
| 1 mM | 2.33 mL | 11.66 mL | 23.31 mL |
| 5 mM | 0.47 mL | 2.33 mL | 4.66 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2