AG 957
目录号: A13589
p210 tyrosine kinase 抑制剂
Tyrphostin AG 957 是一种强效的酪氨酸激酶抑制剂。它选择性地阻断人类 p210bcr-abl 的酪氨酸激酶活性(Ki = 750 nM),相比之下对 p140c-abl 的抑制作用较弱(Ki = 10 μM)。
Discription | Tyrphostin AG 957 is a potent tyrosine kinase inhibitor. Selectively blocks the tyrosine kinase activity of human p210bcr-abl (Ki = 750 nM) over p140c-abl (Ki = 10 μM). | |||||
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Cell Research |
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目录号 | A13589 |
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分子式 | C15H15NO4 |
分子量 | 273.28 |
CAS号 | 140674-76-6 |
SMILES | COC(=O)C1=CC=C(C=C1)NCC2=C(C=CC(=C2)O)O |
其他名称 | Lavendustin C Analog, AG-957, AG957 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2