Trusted by 10,000+ Scientists since 2006
微信关注
申请试用装

AGI-6780

IDH2 R140Q 抑制剂

0 Customer Reviews
产品目录号: A12903

库存状态:中国现货中国现货

产品名 目录号 价格 数量
AGI-6780 5mg A12903-5
¥ 800.00
AGI-6780 10mg A12903-10
¥ 1,400.00
AGI-6780 25mg A12903-25
¥ 2,800.00
AGI-6780 50mg A12903-50
¥ 5,000.00
AGI-6780 10mM * 1mL in DMSO A12903-10mM-D
¥ 1,360.00

产品仅用于研究,不针对患者销售,望谅解.

产品简介

AGI-6780 is a potent, selective inhibitor of mutant IDH2 with an IC50 value of 23 nM.

AGI-6780

双击上述图片即可查看完整大小

缩小
放大

更多视图

顾客使用 Adooq 产品发表的高质量科研文献

Chemical Information

目录号 A12903
Mechanism of action Inhibitor
分子量 481.5
化学分子式 C21H18F3N3O3S
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 1432660-47-3
Synonyms AGI6780
SMILES code C1CC1NS(=O)(=O)C2=CC(=C(C=C2)C3=CSC=C3)NC(=O)NC4=CC=CC(=C4)C(F)(F)F
化学名称 N-?cyclopropyl-?4-?(3-?thienyl)-?3-?[[[[3-?(trifluoromethyl)phenyl]amino]carbonyl]amino]-?benzenesulfonamide

生物活性

Description
AGI-6780 is a potent, selective inhibitor of mutant IDH2 with an IC50 value of 23 nM.
Targets
IDH2 R140Q mutant
23 nM

溶解性

Solubility (25°C)* In vitro DMSO 96 mg/mL (199.37 mM)
Water <1 mg/mL (<1 mM)
Ethanol 96 mg/mL (199.37 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.77 mL 103.84 mL 207.68mL
0.5 mM 4.15 mL 20.77 mL 41.54 mL
1 mM 2.08 mL 10.38 mL 20.77 mL
5 mM 0.42 mL 2.08 mL 4.15 mL

*The above data is based on the productmolecular weight 481.5. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

View Related Products By Research Topics

Ordering online

To place an order online, simply browse to the product you are interested in and click on the 'Add to Cart' button. To complete this process, you will need to confirm the size and quantity of the products that you require.

To complete an order you will need to register using our simple online registration process. We do not share your contact details with any third parties.

When you are ready to check out simply enter your PO number to complete the ordering process. Please ensure that you send us a copy of your PO by fax or email afterwards.  We will then liaise with you or your purchasing department to confirm the order.

Found your products but not ready to order?

Why not use our WishList feature to store lists of products? This convenient feature allows you to manage lists, append notes to products and share lists with co-workers or colleagues.

Ordering offline

You can email or fax us your purchase order and we will place the order for you. You can also phone us to place the order.  Our contact details are:

We require the following information to process your order:
  • The catalog number for each product. 
  • Your email address or fax number. 
  • Your name and telephone number. 
  • Shipping address and billing address.
  • Purchase order numbers.

产品标签

其他人对该产品使用了下列标签:

使用空格分隔标签。使用单引号(')标注词组。


Keywords:购买 AGI-6780 | AGI-6780 供应商 | 订购 AGI-6780 | AGI-6780 价格 | AGI-6780 生产商 | 订单 AGI-6780 | AGI-6780 代理商 | 购买 1432660-47-3| 1432660-47-3 供应商 | 订购 1432660-47-3 | 1432660-47-3 价格 | 1432660-47-3 生产商 | 订单 1432660-47-3 | 1432660-47-3 代理商|buy AGI-6780 | AGI-6780 Supplier | purchase AGI-6780 | AGI-6780 cost | AGI-6780 manufacturer | order AGI-6780 | AGI-6780 distributor | buy 1432660-47-3| 1432660-47-3 Supplier | purchase 1432660-47-3 | 1432660-47-3 cost | 1432660-47-3 manufacturer | order 1432660-47-3 | 1432660-47-3 distributor