Agomelatine

Name: Agomelatine
SKU: A10048

目录号: A10048

5-HT Receptor 拮抗剂

Agomelatine Chemical Structure

CAS NO. 138112-76-2

Agomelatine是一种褪黑素激动剂（MT1和MT2受体）和5-HT2C拮抗剂。

库存：现货

规格	价格	数量
10 mg	￥ 400.00
50 mg	￥ 1,500.00
100 mg	￥ 2,500.00
200 mg	￥ 4,500.00
10mM * 1mL in DMSO	￥ 690.00

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生物活性

Agomelatine是一种褪黑素激动剂（MT1和MT2受体）和5-HT2C拮抗剂。

靶点信息

5-HT2C

溶解度 *

In vitro	DMSO	48 mg/mL (197.28 mM)
	Water	Insoluble
	Ethanol	48 mg/mL (197.28 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	41.1 mL	205.51 mL	411.02 mL
0.5 mM	8.22 mL	41.1 mL	82.2 mL
1 mM	4.11 mL	20.55 mL	41.1 mL
5 mM	0.82 mL	4.11 mL	8.22 mL

*The above data is based on the productmolecular weight 243.3 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A10048
作用机制	Antagonist (拮抗剂)
M. Wt	243.3
Formula	C15H17NO2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	138112-76-2
Synonyms	Valdoxan, Melitor, Thymanax
SMILES	CC(=O)NCCC1=CC=CC2=C1C=C(C=C2)OC