AM-4668
目录号: A21778
GPR40 激动剂
AM-4668 是一种用于治疗2型糖尿病的 GPR40 激动剂。在 A9 细胞(GPR40 IP3 检测)中的 EC50 为 3.6 nM,在 CHO 细胞(GPR40 aequorin 检测)中的 EC50 为 36 nM。
Discription | AM-4668 is a GPR40 agonist for type 2 diabetes. EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively. | |||||
---|---|---|---|---|---|---|
Cell Research |
|
目录号 | A21778 |
---|---|
分子式 | C24H19F3N2O4S |
分子量 | 488.48 |
CAS号 | 1011531-27-3 |
SMILES | OC(C[C@H](C1=NOC=C1)C(C=C2)=CC=C2OCC(S3)=C(C)N=C3C4=CC=C(C(F)(F)F)C=C4)=O |
其他名称 | AM 4668; AM4668 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2