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CB1 receptor 拮抗剂

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产品目录号: A12914


产品名 目录号 价格 数量
AM251 10mg A12914-10
¥ 650.00
AM251 25mg A12914-25
¥ 1,250.00
AM251 50mg A12914-50
¥ 2,400.00
AM251 100mg A12914-100
¥ 4,000.00
AM251 10mM * 1mL in DMSO A12914-10mM-D
¥ 1,060.00



AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors.





顾客使用 Adooq 产品发表的高质量科研文献

Chemical Information

目录号 A12914
Mechanism of action Antagonist
分子量 555.24
化学分子式 C22H21Cl2IN4O
Solubility DMSO
纯度 >98%
储存方式 at -20°C 2 years
CAS No. 183232-66-8
Synonyms AM 251, AM-251
SMILES code CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I
化学名称 N-(Piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide


AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors.


Solubility (25°C) * In vitro DMSO 40 mg/mL (72.04 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 8 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.


Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.01 mL 90.05 mL 180.1mL
0.5 mM 3.6 mL 18.01 mL 36.02 mL
1 mM 1.8 mL 9.01 mL 18.01 mL
5 mM 0.36 mL 1.8 mL 3.6 mL

*The above data is based on the productmolecular weight 555.24. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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