AM251

AM251 Chemical Structure

CAS NO. 183232-66-8

AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors.

库存: 现货

规格 价格 数量
10 mg
¥ 650.00
25 mg
¥ 1,250.00
50 mg
¥ 2,400.00
100 mg
¥ 4,000.00
10mM * 1mL in DMSO
¥ 1,060.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.

详情

AM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors.
Targets
CB1
In vitro (25°C) DMSO 40 mg/mL (72.04 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 8 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.01 mL 90.05 mL 180.1 mL
0.5 mM 3.6 mL 18.01 mL 36.02 mL
1 mM 1.8 mL 9.01 mL 18.01 mL
5 mM 0.36 mL 1.8 mL 3.6 mL

*The above data is based on the productmolecular weight 555.24. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

目录号 A12914
MECHANISM OF ACTION Antagonist
M. Wt 555.24
Formula C22H21Cl2IN4O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 183232-66-8
Synonyms AM 251, AM-251
SMILES CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I

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