Ambrisentan (BSF 208075)

Name: Ambrisentan (BSF 208075)
SKU: A11291

目录号: A11291

EndothelinA receptor 拮抗剂

Product Citations (3)

Ambrisentan (BSF 208075) Chemical Structure

CAS NO. 177036-94-1

Ambrisentan (BSF 208075)充当内皮素受体拮抗剂，对A型内皮素受体（ETA）具有选择性。

库存：现货

规格	价格	数量
5 mg	￥ 500.00
10 mg	￥ 600.00
25 mg	￥ 1,100.00
50 mg	￥ 1,900.00
10mM * 1mL in DMSO	￥ 500.00

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生物活性

Ambrisentan (BSF 208075)充当内皮素受体拮抗剂，对A型内皮素受体（ETA）具有选择性。

靶点信息

ET-A

溶解度 *

In vitro	DMSO	72 mg/mL (190.26 mM)
	Water	Insoluble
	Ethanol	21 mg/mL (55.49 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	26.43 mL	132.14 mL	264.27 mL
0.5 mM	5.29 mL	26.43 mL	52.85 mL
1 mM	2.64 mL	13.21 mL	26.43 mL
5 mM	0.53 mL	2.64 mL	5.29 mL

*The above data is based on the productmolecular weight 378.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A11291
作用机制	Antagonist (拮抗剂)
M. Wt	378.4
Formula	C22H22N2O4
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	177036-94-1
Synonyms	BSF 208075,
SMILES	CC1=CC(=NC(=N1)O[C@H](C(=O)O)C(C2=CC=CC=C2)(C3=CC=CC=C3)OC)C