AMG 837
FFAR1/GPR40 激动剂
FFAR1/GPR40 激动剂
Discription | AMG 837 is a potent GPR40 agonist (EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. |
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Cell Research |
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目录号 | A21160 |
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分子式 | C26H21F3O3 |
分子量 | 438.44 |
CAS号 | 865231-46-5 |
SMILES | OC(C[C@H](C#CC)C1=CC=C(C=C1)OCC2=CC=CC(C3=CC=C(C(F)(F)F)C=C3)=C2)=O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2