AP5
目录号: A20042
AP5 表现出对 GPR40 受体的强效和选择性激动作用,并对内源性配体具有正向的异构调节作用(AgoPAM)。AP5 在针对 GPR40 受体的大鼠 hIP1 EC50 测试中显示出 0.49±0.28 nM 的结果。
Discription | AP5 exhibits potent and selective agonism for the GPR40 receptor with positive allosteric modulation of endogenous ligands (AgoPAM). AP5 demonstrates a rat hIP1 EC50 of 0.49±0.28 nM against the GPR40 receptor. |
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目录号 | A20042 |
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分子式 | C28H28FNO4 |
分子量 | 461.52 |
CAS号 | 1623194-37-5 |
SMILES | FC1=CC(C2=CC(OC)=NC=C2)=CC=C1[C@@H]3CCC(C=CC([C@H](C4CC4)[C@H](C)C(O)=O)=C5)=C5O3 |
其他名称 | AP 5, AP-5 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2