Apatinib (YN968D1)

Name: Apatinib (YN968D1)
SKU: A11407
Price: 700 CNY
Rating: 5 (2 reviews)

目录号: A11407

VEGFR 抑制剂

2 篇发表文献

Apatinib（YN968D1）是一种酪氨酸激酶抑制剂，它选择性地抑制血管内皮生长因子受体-2（VEGFR2，也称为KDR），从而抑制VEGF介导的内皮细胞迁移和增殖，阻断肿瘤组织中新血管的形成。

Skip to the end of the images gallery

Skip to the beginning of the images gallery

Grouped product items
规格	价格	库存
5mg	¥700.00	现货
10mg	¥1,050.00	现货
50mg	¥2,450.00	现货
100mg	¥3,150.00	现货
*10mM 1mL in DMSO**	¥770.00	现货
更大包装	更多折扣

大包装询价

Notify me when the price drops

全国免运费, 顺丰次日达

重要通知：仅供研究使用。我们不向患者销售。

Data Sheet

SDS

Other Forms of Apatinib (YN968D1)

Apatinib mesylate

顾客使用 Adooq 产品发表的高质量科研文献

Adooq用户使用Apatinib (YN968D1)发表的2篇文献

Wonjin Park, .et al. , Biomed Pharmacother, 2021, Feb;134:111110 PMID: 33338749

Majid Momeny, .et al. , Sci Rep, 2017, 7: 45954 PMID: 28383032

生物活性

Discription

Apatinib (YN968D1) is a tyrosine kinase inhibitor that selectively inhibits the vascular endothelial growth factor receptor-2 (VEGFR2, also known as KDR) that inhibits VEGF-mediated endothelial cell migration and proliferation thus blocking new blood vessel formation in tumor tissue.

Targets

Target	Value

产品信息

目录号	A11407
分子式	C25H27N5O4S
分子量	493.6
CAS号	811803-05-1
SMILES	CS(=O)(=O)O.C1CCC(C1)(C#N)C2=CC=C(C=C2)NC(=O)C3=C(N=CC=C3)NCC4=CC=NC=C4
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	77 mg/mL (193.72 mM)
	Water	Insoluble
	Ethanol	10 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	20.26 mL	101.3 mL	202.59 mL
0.5 mM	4.05 mL	20.26 mL	40.52 mL
1 mM	2.03 mL	10.13 mL	20.26 mL
5 mM	0.41 mL	2.03 mL	4.05 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

Calculate Reset

* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

Keywords: 购买 Apatinib (YN968D1) | Apatinib (YN968D1) 供应商 | Apatinib (YN968D1) 花费 | Apatinib (YN968D1) 生产商 | 订购 Apatinib (YN968D1) | Apatinib (YN968D1) 代理商 | 购买 811803-05-1 | 811803-05-1 供应商 | 811803-05-1 花费 | 811803-05-1 生产商 | 订购 811803-05-1 | 811803-05-1 代理商