APD668
目录号: A14342
GPR119 激动剂
APD668 是一种强效的 GPR119 激动剂,其 EC50 分别为 2.7 nM 和 33 nM,针对 hGPR119 和 ratGPR119。
Discription | APD668 is a potent GPR119 agonist with EC50 of 2.7 nM and 33 nM for hGPR119 and ratGPR119 respectively. | ||
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Targets |
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目录号 | A14342 |
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分子式 | C21H24FN5O5S |
分子量 | 477.51 |
CAS号 | 832714-46-2 |
SMILES | CC(C)OC(=O)N1CCC(CC1)OC2=NC=NC3=C2C=NN3C4=C(C=C(C=C4)S(=O)(=O)C)F |
其他名称 | APD 668, APD-668, JNJ-28630368, JNJ28630368, JNJ 28630368 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 86 mg/mL (180.1 mM) | |
Water | Insoluble | ||
Ethanol | 2 mg/mL (4.18 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 20.94 mL | 104.71 mL | 209.42 mL |
0.5 mM | 4.19 mL | 20.94 mL | 41.88 mL |
1 mM | 2.09 mL | 10.47 mL | 20.94 mL |
5 mM | 0.42 mL | 2.09 mL | 4.19 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2